IndraLab

Statements


KCNH2 binds AZA1. 1 / 1
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"Relative to vehicle controls, hERG binding by AZA1, AZA2, and AZA3 (10 muM) was reduced to 19.7 +/- 1.4% (n = 2), 22.3 +/- 1.0% (n = 3), and 29.3 +/- 1.6% (n = 3) with IC 50 values of 2.1 muM, 2.6 muM, and 6.6 muM; respectively (XREF_TABLE)."