IndraLab

Statements


E-4031 K inhibits KCNH2. 1 / 1
| 1

reach
"In CHO cells, HERG channels were strongly blocked by E-4031 K i = 8.8 +/- 0.8 nM; again, channels formed with hMiRP1 were ~ 2-fold more sensitive (K i = 4.6 +/- 0.6 nM; n = 6 cells)."