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KCNH2 inhibits antagonist. 1 / 1
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"The in vitro ADMET properties —microsomal metabolism, CYP2D6 inhibition, HSA binding, cell permeability, and hERG inhibition— of the 5-HT 6 R antagonist newly identified herein 7 excluded important pharmacokinetic issues and possible lethal side effects related with cardiac toxicity (see Results section)."